Pyrimido[4,5-d]azepines as potent and selective 5-HT2C receptor agonists: Design, synthesis, and evaluation of PF-3246799 as a treatment for urinary incontinence. Andrews, M. D., Fish, P. V., Blagg, J., Brabham, T. K., Brennan, P. E., Bridgeland, A., Brown, A. D., Bungay, P. J., Conlon, K. M., Edmunds, N. J., af Forselles, K., Gibbons, C. P., Green, M. P., Hanton, G., Holbrook, M., Jessiman, A. S., McIntosh, K., McMurray, G., Nichols, C. L., Root, J. A., Storer, R. I., Sutton, M. R., Ward, R. V., Westbrook, D., & Whitlock, G. A. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 21(9):2715-2720, MAY 1, 2011.
doi  bibtex   
@article{ WOS:000289773300029,
Author = {Andrews, Mark D. and Fish, Paul V. and Blagg, Julian and Brabham,
   Tiffini K. and Brennan, Paul E. and Bridgeland, Alison and Brown, Alan
   D. and Bungay, Peter J. and Conlon, Kelly M. and Edmunds, Nicholas J.
   and af Forselles, Kerry and Gibbons, Colleen P. and Green, Martin P. and
   Hanton, Giles and Holbrook, Mark and Jessiman, Alan S. and McIntosh,
   Karin and McMurray, Gordon and Nichols, Carly L. and Root, James A. and
   Storer, R. Ian and Sutton, Michael R. and Ward, Robin V. and Westbrook,
   Dominique and Whitlock, Gavin A.},
Title = {Pyrimido{[}4,5-d]azepines as potent and selective
   5-HT2C receptor agonists: Design, synthesis, and evaluation
   of PF-3246799 as a treatment for urinary incontinence},
Journal = {BIOORGANIC \& MEDICINAL CHEMISTRY LETTERS},
Year = {2011},
Volume = {21},
Number = {9},
Pages = {2715-2720},
Month = {MAY 1},
DOI = {10.1016/j.bmcl.2010.11.120},
ISSN = {0960-894X},
EISSN = {1464-3405},
ORCID-Numbers = {Brennan, Paul/0000-0002-8950-7646},
Unique-ID = {WOS:000289773300029},
}

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