Discovery of New G-quadruplex Binding Chemotypes. a Ohnmacht, S., Varavipour, E., Nanjunda, R., Pazitna, I., Vita, G. D., Gunaratnam, M., Kumar, A., a Ismail, M., Boykin, D. W, Wilson, W D., & Neidle, S. Chemical communications (Cambridge, England), December, 2013.
doi  abstract   bibtex   
We report here on the discovery and preliminary evaluation of a novel non-macrocyclic low molecular weight quadruplex-stabilizing chemotype. The lead compounds, based on a furan core, show high G-quadruplex stabilisation and selectivity as well as potent in vitro anti-proliferative activity.
@article{Ohnmacht2013,
  title = {Discovery of New {{G-quadruplex}} Binding Chemotypes.},
  author = {a Ohnmacht, Stephan and Varavipour, Ehsan and Nanjunda, Rupesh and Pazitna, Ingrida and Vita, Gloria Di and Gunaratnam, Mekala and Kumar, Arvind and a Ismail, Mohamed and Boykin, David W and Wilson, W David and Neidle, Stephen},
  year = {2013},
  month = dec,
  journal = {Chemical communications (Cambridge, England)},
  eprint = {24302123},
  eprinttype = {pubmed},
  pages = {1--4},
  issn = {1364-548X},
  doi = {10.1039/c3cc48616h},
  abstract = {We report here on the discovery and preliminary evaluation of a novel non-macrocyclic low molecular weight quadruplex-stabilizing chemotype. The lead compounds, based on a furan core, show high G-quadruplex stabilisation and selectivity as well as potent in vitro anti-proliferative activity.},
  pmid = {24302123},
  keywords = {\#nosource}
}

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