@article{
 title = {A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain},
 type = {article},
 year = {2016},
 pages = {2322-2330},
 volume = {7},
 websites = {http://xlink.rsc.org/?DOI=C5SC03115J},
 publisher = {Royal Society of Chemistry},
 id = {7561975c-c867-342f-a40e-65d3f055c4ed},
 created = {2016-02-01T08:09:31.000Z},
 file_attached = {true},
 profile_id = {64f7fb50-d000-335d-a02d-06c5f340a97a},
 last_modified = {2024-05-02T14:04:14.785Z},
 read = {true},
 starred = {true},
 authored = {true},
 confirmed = {true},
 hidden = {false},
 citation_key = {Cox2016},
 folder_uuids = {5358531d-d036-484b-937b-88c0f1ef606b},
 private_publication = {false},
 abstract = {<p> High concentration crystal soaking of poised fragments and one-step elaboration identified compound <bold>17</bold> as an inhibitor of the PHIP(2) bromodomain. </p>},
 bibtype = {article},
 author = {Cox, Oakley B. and Krojer, Tobias and Collins, Patrick and Monteiro, Octovia and Talon, Romain and Bradley, Anthony and Fedorov, Oleg and Amin, Jahangir and Marsden, Brian D. and Spencer, John and Von Delft, Frank and Brennan, Paul E.},
 doi = {10.1039/c5sc03115j},
 journal = {Chemical Science},
 number = {3}
}

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