A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain. Cox, O. B., Krojer, T., Collins, P., Monteiro, O., Talon, R., Bradley, A., Fedorov, O., Amin, J., Marsden, B. D., Spencer, J., von Delft, F., & Brennan, P. E. CHEMICAL SCIENCE, 7(3):2322-2330, 2016.
doi  bibtex   
@article{ WOS:000371021900087,
Author = {Cox, Oakley B. and Krojer, Tobias and Collins, Patrick and Monteiro,
   Octovia and Talon, Romain and Bradley, Anthony and Fedorov, Oleg and
   Amin, Jahangir and Marsden, Brian D. and Spencer, John and von Delft,
   Frank and Brennan, Paul E.},
Title = {A poised fragment library enables rapid synthetic expansion yielding the
   first reported inhibitors of PHIP(2), an atypical bromodomain},
Journal = {CHEMICAL SCIENCE},
Year = {2016},
Volume = {7},
Number = {3},
Pages = {2322-2330},
DOI = {10.1039/c5sc03115j},
ISSN = {2041-6520},
EISSN = {2041-6539},
ResearcherID-Numbers = {SPENCER, John/P-5492-2019
   Krojer, Tobias/ABE-3829-2021
   Collins, Patrick/C-7960-2016
   Spencer, John/C-2156-2008
   },
ORCID-Numbers = {Talon, Romain/0000-0003-1123-7241
   Brennan, Paul/0000-0002-8950-7646
   Collins, Patrick/0000-0002-6265-9922
   von Delft, Frank/0000-0003-0378-0017
   Spencer, John/0000-0001-5231-8836
   Krojer, Tobias/0000-0003-0661-0814},
Unique-ID = {WOS:000371021900087},
}

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