A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain. Cox, O. B., Krojer, T., Collins, P., Monteiro, O., Talon, R., Bradley, A., Fedorov, O., Amin, J., Marsden, B. D., Spencer, J., von Delft, F., & Brennan, P. E. CHEMICAL SCIENCE, 7(3):2322-2330, 2016. doi bibtex @article{ WOS:000371021900087,
Author = {Cox, Oakley B. and Krojer, Tobias and Collins, Patrick and Monteiro,
Octovia and Talon, Romain and Bradley, Anthony and Fedorov, Oleg and
Amin, Jahangir and Marsden, Brian D. and Spencer, John and von Delft,
Frank and Brennan, Paul E.},
Title = {A poised fragment library enables rapid synthetic expansion yielding the
first reported inhibitors of PHIP(2), an atypical bromodomain},
Journal = {CHEMICAL SCIENCE},
Year = {2016},
Volume = {7},
Number = {3},
Pages = {2322-2330},
DOI = {10.1039/c5sc03115j},
ISSN = {2041-6520},
EISSN = {2041-6539},
ResearcherID-Numbers = {SPENCER, John/P-5492-2019
Krojer, Tobias/ABE-3829-2021
Collins, Patrick/C-7960-2016
Spencer, John/C-2156-2008
},
ORCID-Numbers = {Talon, Romain/0000-0003-1123-7241
Brennan, Paul/0000-0002-8950-7646
Collins, Patrick/0000-0002-6265-9922
von Delft, Frank/0000-0003-0378-0017
Spencer, John/0000-0001-5231-8836
Krojer, Tobias/0000-0003-0661-0814},
Unique-ID = {WOS:000371021900087},
}
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