Discovery of a Series of 5-Azaquinazolines as Orally Efficacious IRAK4 Inhibitors Targeting MyD88 $^{\textrm{{L265P}}}$ Mutant Diffuse Large B Cell Lymphoma. Degorce, S. L., Anjum, R., Bloecher, A., Carbajo, R. J., Dillman, K. S., Drew, L., Halsall, C. T., Lenz, E. M., Lindsay, N. A., Mayo, M. F., Pink, J. H., Robb, G. R., Rosen, A., Scott, J. S., & Xue, Y. Journal of Medicinal Chemistry, 62(21):9918–9930, November, 2019. ![Discovery of a Series of 5-Azaquinazolines as Orally Efficacious IRAK4 Inhibitors Targeting MyD88 $^{\textrm{{L265P}}}$ Mutant Diffuse Large B Cell Lymphoma [link]](https://bibbase.org/img/filetypes/link.svg "link")
Paper doi bibtex @article{degorce_discovery_2019,
title = {Discovery of a {Series} of 5-{Azaquinazolines} as {Orally} {Efficacious} {IRAK4} {Inhibitors} {Targeting} {MyD88} $^{\textrm{{L265P}}}$ {Mutant} {Diffuse} {Large} {B} {Cell} {Lymphoma}},
volume = {62},
issn = {0022-2623, 1520-4804},
url = {https://pubs.acs.org/doi/10.1021/acs.jmedchem.9b01346},
doi = {10.1021/acs.jmedchem.9b01346},
language = {en},
number = {21},
urldate = {2023-09-26},
journal = {Journal of Medicinal Chemistry},
author = {Degorce, Sébastien L. and Anjum, Rana and Bloecher, Andrew and Carbajo, Rodrigo J. and Dillman, Keith S. and Drew, Lisa and Halsall, Christopher T. and Lenz, Eva M. and Lindsay, Nicola A. and Mayo, Michele F. and Pink, Jennifer H. and Robb, Graeme R. and Rosen, Alan and Scott, James S. and Xue, Yafeng},
month = nov,
year = {2019},
pages = {9918--9930},
}
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