@article{
 title = {Optimisation of a triazolopyridine based histone demethylase inhibitor yields a potent and selective KDM2A (FBXL11) inhibitor},
 type = {article},
 year = {2014},
 pages = {1879-1886},
 volume = {5},
 websites = {http://dx.doi.org/10.1039/C4MD00291A,http://pubs.rsc.org/en/content/articlepdf/2014/md/c4md00291a},
 publisher = {The Royal Society of Chemistry},
 id = {d42854e0-accf-3fb1-a2e2-2d8ccbd34af4},
 created = {2015-10-01T17:18:05.000Z},
 file_attached = {true},
 profile_id = {64f7fb50-d000-335d-a02d-06c5f340a97a},
 last_modified = {2018-09-03T10:20:45.992Z},
 read = {true},
 starred = {true},
 authored = {true},
 confirmed = {true},
 hidden = {false},
 citation_key = {England2014},
 source_type = {Journal Article},
 private_publication = {false},
 abstract = {<p> Compound <bold>35</bold> is a potent and selective triazolopyridine inhibitor of the lysine demethylase KDM2A (pIC <sub>50</sub> 7.2). </p>},
 bibtype = {article},
 author = {England, Katherine S. and Tumber, Anthony and Krojer, Tobias and Scozzafava, Giuseppe and Ng, Stanley S. and Daniel, Michelle and Szykowska, Aleksandra and Che, Kahing and Von Delft, Frank and Burgess-Brown, Nicola A. and Kawamura, Akane and Schofield, Christopher J. and Brennan, Paul E.},
 doi = {10.1039/c4md00291a},
 journal = {MedChemComm},
 number = {12}
}

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