@article{ WOS:000311461500035,
Author = {Fish, Paul V. and Filippakopoulos, Panagis and Bish, Gerwyn and Brennan,
   Paul E. and Bunnage, Mark E. and Cook, Andrew S. and Federov, Oleg and
   Gerstenberger, Brian S. and Jones, Hannah and Knapp, Stefan and Marsden,
   Brian and Nocka, Karl and Owen, Dafydd R. and Philpott, Martin and
   Picaud, Sarah and Primiano, Michael J. and Ralph, Michael J. and
   Sciammetta, Nunzio and Trzupek, John D.},
Title = {Identification of a Chemical Probe for Bromo and Extra C-Terminal
   Bromodomain Inhibition through Optimization of a Fragment-Derived Hit},
Journal = {JOURNAL OF MEDICINAL CHEMISTRY},
Year = {2012},
Volume = {55},
Number = {22},
Pages = {9831-9837},
Month = {NOV 22},
DOI = {10.1021/jm3010515},
ISSN = {0022-2623},
EISSN = {1520-4804},
ResearcherID-Numbers = {Brown, Tom/A-6655-2010
   Primiano, Michael/HPD-4541-2023
   Jones, Hannah/AAM-5162-2020
   Knapp, Stefan/AAG-2347-2019
   },
ORCID-Numbers = {Filippakopoulos, Panagis/0000-0002-1515-1317
   Knapp, Stefan/0000-0001-5995-6494
   Philpott, Martin/0000-0003-3632-0084
   Bunnage, Mark/0009-0002-6063-8041},
Unique-ID = {WOS:000311461500035},
}

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D."],"year":2012,"bibtype":"article","biburl":"https://bibbase.org/network/files/HECPruWhe6gDg5ZWN","bibdata":{"bibtype":"article","type":"article","author":[{"propositions":[],"lastnames":["Fish"],"firstnames":["Paul","V."],"suffixes":[]},{"propositions":[],"lastnames":["Filippakopoulos"],"firstnames":["Panagis"],"suffixes":[]},{"propositions":[],"lastnames":["Bish"],"firstnames":["Gerwyn"],"suffixes":[]},{"propositions":[],"lastnames":["Brennan"],"firstnames":["Paul","E."],"suffixes":[]},{"propositions":[],"lastnames":["Bunnage"],"firstnames":["Mark","E."],"suffixes":[]},{"propositions":[],"lastnames":["Cook"],"firstnames":["Andrew","S."],"suffixes":[]},{"propositions":[],"lastnames":["Federov"],"firstnames":["Oleg"],"suffixes":[]},{"propositions":[],"lastnames":["Gerstenberger"],"firstnames":["Brian","S."],"suffixes":[]},{"propositions":[],"lastnames":["Jones"],"firstnames":["Hannah"],"suffixes":[]},{"propositions":[],"lastnames":["Knapp"],"firstnames":["Stefan"],"suffixes":[]},{"propositions":[],"lastnames":["Marsden"],"firstnames":["Brian"],"suffixes":[]},{"propositions":[],"lastnames":["Nocka"],"firstnames":["Karl"],"suffixes":[]},{"propositions":[],"lastnames":["Owen"],"firstnames":["Dafydd","R."],"suffixes":[]},{"propositions":[],"lastnames":["Philpott"],"firstnames":["Martin"],"suffixes":[]},{"propositions":[],"lastnames":["Picaud"],"firstnames":["Sarah"],"suffixes":[]},{"propositions":[],"lastnames":["Primiano"],"firstnames":["Michael","J."],"suffixes":[]},{"propositions":[],"lastnames":["Ralph"],"firstnames":["Michael","J."],"suffixes":[]},{"propositions":[],"lastnames":["Sciammetta"],"firstnames":["Nunzio"],"suffixes":[]},{"propositions":[],"lastnames":["Trzupek"],"firstnames":["John","D."],"suffixes":[]}],"title":"Identification of a Chemical Probe for Bromo and Extra C-Terminal Bromodomain Inhibition through Optimization of a Fragment-Derived Hit","journal":"JOURNAL OF MEDICINAL CHEMISTRY","year":"2012","volume":"55","number":"22","pages":"9831-9837","month":"NOV 22","doi":"10.1021/jm3010515","issn":"0022-2623","eissn":"1520-4804","researcherid-numbers":"Brown, Tom/A-6655-2010 Primiano, Michael/HPD-4541-2023 Jones, Hannah/AAM-5162-2020 Knapp, Stefan/AAG-2347-2019 ","orcid-numbers":"Filippakopoulos, Panagis/0000-0002-1515-1317 Knapp, Stefan/0000-0001-5995-6494 Philpott, Martin/0000-0003-3632-0084 Bunnage, Mark/0009-0002-6063-8041","unique-id":"WOS:000311461500035","bibtex":"@article{ WOS:000311461500035,\nAuthor = {Fish, Paul V. and Filippakopoulos, Panagis and Bish, Gerwyn and Brennan,\n Paul E. and Bunnage, Mark E. and Cook, Andrew S. and Federov, Oleg and\n Gerstenberger, Brian S. and Jones, Hannah and Knapp, Stefan and Marsden,\n Brian and Nocka, Karl and Owen, Dafydd R. and Philpott, Martin and\n Picaud, Sarah and Primiano, Michael J. and Ralph, Michael J. and\n Sciammetta, Nunzio and Trzupek, John D.},\nTitle = {Identification of a Chemical Probe for Bromo and Extra C-Terminal\n Bromodomain Inhibition through Optimization of a Fragment-Derived Hit},\nJournal = {JOURNAL OF MEDICINAL CHEMISTRY},\nYear = {2012},\nVolume = {55},\nNumber = {22},\nPages = {9831-9837},\nMonth = {NOV 22},\nDOI = {10.1021/jm3010515},\nISSN = {0022-2623},\nEISSN = {1520-4804},\nResearcherID-Numbers = {Brown, Tom/A-6655-2010\n Primiano, Michael/HPD-4541-2023\n Jones, Hannah/AAM-5162-2020\n Knapp, Stefan/AAG-2347-2019\n },\nORCID-Numbers = {Filippakopoulos, Panagis/0000-0002-1515-1317\n Knapp, Stefan/0000-0001-5995-6494\n Philpott, Martin/0000-0003-3632-0084\n Bunnage, Mark/0009-0002-6063-8041},\nUnique-ID = {WOS:000311461500035},\n}\n\n","author_short":["Fish, P. 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