Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit. Gerstenberger, B. S., Trzupek, J. D., Tallant, C., Fedorov, O., Filippakopoulos, P., Brennan, P. E., Fedele, V., Martin, S., Picaud, S., Rogers, C., Parikh, M., Taylor, A., Samas, B., O'Mahony, A., Berg, E., Pallares, G., Torrey, A. D., Treiber, D. K., Samardjiev, I. J., Nasipak, B. T., Padilla-Benavides, T., Wu, Q., Imbalzano, A. N., Nickerson, J. A., Bunnage, M. E., Muller, S., Knapp, S., & Owen, D. R. JOURNAL OF MEDICINAL CHEMISTRY, 59(10):4800-4811, MAY 26, 2016. doi bibtex @article{ WOS:000376840600030,
Author = {Gerstenberger, Brian S. and Trzupek, John D. and Tallant, Cynthia and
Fedorov, Oleg and Filippakopoulos, Panagis and Brennan, Paul E. and
Fedele, Vita and Martin, Sarah and Picaud, Sarah and Rogers, Catherine
and Parikh, Mihir and Taylor, Alexandria and Samas, Brian and O'Mahony,
Alison and Berg, Ellen and Pallares, Gabriel and Torrey, Adam D. and
Treiber, Daniel K. and Samardjiev, Ivan J. and Nasipak, Brian T. and
Padilla-Benavides, Teresita and Wu, Qiong and Imbalzano, Anthony N. and
Nickerson, Jeffrey A. and Bunnage, Mark E. and Muller, Susanne and
Knapp, Stefan and Owen, Dafydd R.},
Title = {Identification of a Chemical Probe for Family VIII Bromodomains through
Optimization of a Fragment Hit},
Journal = {JOURNAL OF MEDICINAL CHEMISTRY},
Year = {2016},
Volume = {59},
Number = {10},
Pages = {4800-4811},
Month = {MAY 26},
DOI = {10.1021/acs.jmedchem.6b00012},
ISSN = {0022-2623},
EISSN = {1520-4804},
ResearcherID-Numbers = {Knapp, Stefan/AAG-2347-2019
Berg, Ellen/T-8827-2019
Fedorov, Oleg/B-6412-2014
Berg, Ellen/D-9076-2014
PADILLA-BENAVIDES, TERESITA/K-1968-2012
},
ORCID-Numbers = {Brennan, Paul/0000-0002-8950-7646
Berg, Ellen/0000-0001-5149-6665
Filippakopoulos, Panagis/0000-0002-1515-1317
Knapp, Stefan/0000-0001-5995-6494
Bunnage, Mark/0009-0002-6063-8041
PADILLA-BENAVIDES, TERESITA/0000-0002-4624-0822
Tallant, Cynthia/0000-0001-5645-435X
Muller-Knapp, Susanne/0000-0003-2402-4157},
Unique-ID = {WOS:000376840600030},
}
Downloads: 0
{"_id":"R8iA9jP37yX2r34nk","bibbaseid":"gerstenberger-trzupek-tallant-fedorov-filippakopoulos-brennan-fedele-martin-etal-identificationofachemicalprobeforfamilyviiibromodomainsthroughoptimizationofafragmenthit-2016","downloads":0,"creationDate":"2018-08-31T13:28:42.414Z","title":"Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit","author_short":["Gerstenberger, B. S.","Trzupek, J. D.","Tallant, C.","Fedorov, O.","Filippakopoulos, P.","Brennan, P. E.","Fedele, V.","Martin, S.","Picaud, S.","Rogers, C.","Parikh, M.","Taylor, A.","Samas, B.","O'Mahony, A.","Berg, E.","Pallares, G.","Torrey, A. D.","Treiber, D. K.","Samardjiev, I. J.","Nasipak, B. T.","Padilla-Benavides, T.","Wu, Q.","Imbalzano, A. N.","Nickerson, J. A.","Bunnage, M. E.","Muller, S.","Knapp, S.","Owen, D. R."],"year":2016,"bibtype":"article","biburl":"https://bibbase.org/network/files/HECPruWhe6gDg5ZWN","bibdata":{"bibtype":"article","type":"article","author":[{"propositions":[],"lastnames":["Gerstenberger"],"firstnames":["Brian","S."],"suffixes":[]},{"propositions":[],"lastnames":["Trzupek"],"firstnames":["John","D."],"suffixes":[]},{"propositions":[],"lastnames":["Tallant"],"firstnames":["Cynthia"],"suffixes":[]},{"propositions":[],"lastnames":["Fedorov"],"firstnames":["Oleg"],"suffixes":[]},{"propositions":[],"lastnames":["Filippakopoulos"],"firstnames":["Panagis"],"suffixes":[]},{"propositions":[],"lastnames":["Brennan"],"firstnames":["Paul","E."],"suffixes":[]},{"propositions":[],"lastnames":["Fedele"],"firstnames":["Vita"],"suffixes":[]},{"propositions":[],"lastnames":["Martin"],"firstnames":["Sarah"],"suffixes":[]},{"propositions":[],"lastnames":["Picaud"],"firstnames":["Sarah"],"suffixes":[]},{"propositions":[],"lastnames":["Rogers"],"firstnames":["Catherine"],"suffixes":[]},{"propositions":[],"lastnames":["Parikh"],"firstnames":["Mihir"],"suffixes":[]},{"propositions":[],"lastnames":["Taylor"],"firstnames":["Alexandria"],"suffixes":[]},{"propositions":[],"lastnames":["Samas"],"firstnames":["Brian"],"suffixes":[]},{"propositions":[],"lastnames":["O'Mahony"],"firstnames":["Alison"],"suffixes":[]},{"propositions":[],"lastnames":["Berg"],"firstnames":["Ellen"],"suffixes":[]},{"propositions":[],"lastnames":["Pallares"],"firstnames":["Gabriel"],"suffixes":[]},{"propositions":[],"lastnames":["Torrey"],"firstnames":["Adam","D."],"suffixes":[]},{"propositions":[],"lastnames":["Treiber"],"firstnames":["Daniel","K."],"suffixes":[]},{"propositions":[],"lastnames":["Samardjiev"],"firstnames":["Ivan","J."],"suffixes":[]},{"propositions":[],"lastnames":["Nasipak"],"firstnames":["Brian","T."],"suffixes":[]},{"propositions":[],"lastnames":["Padilla-Benavides"],"firstnames":["Teresita"],"suffixes":[]},{"propositions":[],"lastnames":["Wu"],"firstnames":["Qiong"],"suffixes":[]},{"propositions":[],"lastnames":["Imbalzano"],"firstnames":["Anthony","N."],"suffixes":[]},{"propositions":[],"lastnames":["Nickerson"],"firstnames":["Jeffrey","A."],"suffixes":[]},{"propositions":[],"lastnames":["Bunnage"],"firstnames":["Mark","E."],"suffixes":[]},{"propositions":[],"lastnames":["Muller"],"firstnames":["Susanne"],"suffixes":[]},{"propositions":[],"lastnames":["Knapp"],"firstnames":["Stefan"],"suffixes":[]},{"propositions":[],"lastnames":["Owen"],"firstnames":["Dafydd","R."],"suffixes":[]}],"title":"Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit","journal":"JOURNAL OF MEDICINAL CHEMISTRY","year":"2016","volume":"59","number":"10","pages":"4800-4811","month":"MAY 26","doi":"10.1021/acs.jmedchem.6b00012","issn":"0022-2623","eissn":"1520-4804","researcherid-numbers":"Knapp, Stefan/AAG-2347-2019 Berg, Ellen/T-8827-2019 Fedorov, Oleg/B-6412-2014 Berg, Ellen/D-9076-2014 PADILLA-BENAVIDES, TERESITA/K-1968-2012 ","orcid-numbers":"Brennan, Paul/0000-0002-8950-7646 Berg, Ellen/0000-0001-5149-6665 Filippakopoulos, Panagis/0000-0002-1515-1317 Knapp, Stefan/0000-0001-5995-6494 Bunnage, Mark/0009-0002-6063-8041 PADILLA-BENAVIDES, TERESITA/0000-0002-4624-0822 Tallant, Cynthia/0000-0001-5645-435X Muller-Knapp, Susanne/0000-0003-2402-4157","unique-id":"WOS:000376840600030","bibtex":"@article{ WOS:000376840600030,\nAuthor = {Gerstenberger, Brian S. and Trzupek, John D. and Tallant, Cynthia and\n Fedorov, Oleg and Filippakopoulos, Panagis and Brennan, Paul E. and\n Fedele, Vita and Martin, Sarah and Picaud, Sarah and Rogers, Catherine\n and Parikh, Mihir and Taylor, Alexandria and Samas, Brian and O'Mahony,\n Alison and Berg, Ellen and Pallares, Gabriel and Torrey, Adam D. and\n Treiber, Daniel K. and Samardjiev, Ivan J. and Nasipak, Brian T. and\n Padilla-Benavides, Teresita and Wu, Qiong and Imbalzano, Anthony N. and\n Nickerson, Jeffrey A. and Bunnage, Mark E. and Muller, Susanne and\n Knapp, Stefan and Owen, Dafydd R.},\nTitle = {Identification of a Chemical Probe for Family VIII Bromodomains through\n Optimization of a Fragment Hit},\nJournal = {JOURNAL OF MEDICINAL CHEMISTRY},\nYear = {2016},\nVolume = {59},\nNumber = {10},\nPages = {4800-4811},\nMonth = {MAY 26},\nDOI = {10.1021/acs.jmedchem.6b00012},\nISSN = {0022-2623},\nEISSN = {1520-4804},\nResearcherID-Numbers = {Knapp, Stefan/AAG-2347-2019\n Berg, Ellen/T-8827-2019\n Fedorov, Oleg/B-6412-2014\n Berg, Ellen/D-9076-2014\n PADILLA-BENAVIDES, TERESITA/K-1968-2012\n },\nORCID-Numbers = {Brennan, Paul/0000-0002-8950-7646\n Berg, Ellen/0000-0001-5149-6665\n Filippakopoulos, Panagis/0000-0002-1515-1317\n Knapp, Stefan/0000-0001-5995-6494\n Bunnage, Mark/0009-0002-6063-8041\n PADILLA-BENAVIDES, TERESITA/0000-0002-4624-0822\n Tallant, Cynthia/0000-0001-5645-435X\n Muller-Knapp, Susanne/0000-0003-2402-4157},\nUnique-ID = {WOS:000376840600030},\n}\n\n","author_short":["Gerstenberger, B. S.","Trzupek, J. D.","Tallant, C.","Fedorov, O.","Filippakopoulos, P.","Brennan, P. E.","Fedele, V.","Martin, S.","Picaud, S.","Rogers, C.","Parikh, M.","Taylor, A.","Samas, B.","O'Mahony, A.","Berg, E.","Pallares, G.","Torrey, A. D.","Treiber, D. K.","Samardjiev, I. J.","Nasipak, B. T.","Padilla-Benavides, T.","Wu, Q.","Imbalzano, A. N.","Nickerson, J. A.","Bunnage, M. E.","Muller, S.","Knapp, S.","Owen, D. R."],"key":"WOS:000376840600030","id":"WOS:000376840600030","bibbaseid":"gerstenberger-trzupek-tallant-fedorov-filippakopoulos-brennan-fedele-martin-etal-identificationofachemicalprobeforfamilyviiibromodomainsthroughoptimizationofafragmenthit-2016","role":"author","urls":{},"metadata":{"authorlinks":{"brennan, p":"https://lanternfish-chipmunk-64nl.squarespace.com/publications"}},"downloads":0},"search_terms":["identification","chemical","probe","family","viii","bromodomains","through","optimization","fragment","hit","gerstenberger","trzupek","tallant","fedorov","filippakopoulos","brennan","fedele","martin","picaud","rogers","parikh","taylor","samas","o'mahony","berg","pallares","torrey","treiber","samardjiev","nasipak","padilla-benavides","wu","imbalzano","nickerson","bunnage","muller","knapp","owen"],"keywords":[],"authorIDs":["g4JkphGbeNea298iY"],"dataSources":["Pa586au6MYhHM9r97","ya2CyA73rpZseyrZ8","2252seNhipfTmjEBQ","qhzgQBKWKwmm6xY73","NBNKNR2KcNSWDgFcf","4mccB2G6uYe3AhfDs"]}