Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit. Gerstenberger, B. S., Trzupek, J. D., Tallant, C., Fedorov, O., Filippakopoulos, P., Brennan, P. E., Fedele, V., Martin, S., Picaud, S., Rogers, C., Parikh, M., Taylor, A., Samas, B., O'Mahony, A., Berg, E., Pallares, G., Torrey, A. D., Treiber, D. K., Samardjiev, I. J., Nasipak, B. T., Padilla-Benavides, T., Wu, Q., Imbalzano, A. N., Nickerson, J. A., Bunnage, M. E., Muller, S., Knapp, S., & Owen, D. R. JOURNAL OF MEDICINAL CHEMISTRY, 59(10):4800-4811, MAY 26, 2016.
doi  bibtex   
@article{ WOS:000376840600030,
Author = {Gerstenberger, Brian S. and Trzupek, John D. and Tallant, Cynthia and
   Fedorov, Oleg and Filippakopoulos, Panagis and Brennan, Paul E. and
   Fedele, Vita and Martin, Sarah and Picaud, Sarah and Rogers, Catherine
   and Parikh, Mihir and Taylor, Alexandria and Samas, Brian and O'Mahony,
   Alison and Berg, Ellen and Pallares, Gabriel and Torrey, Adam D. and
   Treiber, Daniel K. and Samardjiev, Ivan J. and Nasipak, Brian T. and
   Padilla-Benavides, Teresita and Wu, Qiong and Imbalzano, Anthony N. and
   Nickerson, Jeffrey A. and Bunnage, Mark E. and Muller, Susanne and
   Knapp, Stefan and Owen, Dafydd R.},
Title = {Identification of a Chemical Probe for Family VIII Bromodomains through
   Optimization of a Fragment Hit},
Journal = {JOURNAL OF MEDICINAL CHEMISTRY},
Year = {2016},
Volume = {59},
Number = {10},
Pages = {4800-4811},
Month = {MAY 26},
DOI = {10.1021/acs.jmedchem.6b00012},
ISSN = {0022-2623},
EISSN = {1520-4804},
ResearcherID-Numbers = {Knapp, Stefan/AAG-2347-2019
   Berg, Ellen/T-8827-2019
   Fedorov, Oleg/B-6412-2014
   Berg, Ellen/D-9076-2014
   PADILLA-BENAVIDES, TERESITA/K-1968-2012
   },
ORCID-Numbers = {Brennan, Paul/0000-0002-8950-7646
   Berg, Ellen/0000-0001-5149-6665
   Filippakopoulos, Panagis/0000-0002-1515-1317
   Knapp, Stefan/0000-0001-5995-6494
   Bunnage, Mark/0009-0002-6063-8041
   PADILLA-BENAVIDES, TERESITA/0000-0002-4624-0822
   Tallant, Cynthia/0000-0001-5645-435X
   Muller-Knapp, Susanne/0000-0003-2402-4157},
Unique-ID = {WOS:000376840600030},
}

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