Optimization of 3,5-Dimethylisoxazole Derivatives as Potent Bromodomain Ligands. Hewings, D. S., Fedorov, O., Filippakopoulos, P., Martin, S., Picaud, S., Tumber, A., Wells, C., Olcina, M. M., Freeman, K., Gill, A., Ritchie, A. J., Sheppard, D. W., Russell, A. J., Hammond, E. M., Knapp, S., Brennan, P. E., & Conway, S. J. JOURNAL OF MEDICINAL CHEMISTRY, 56(8):3217-3227, APR 25, 2013. doi bibtex @article{ WOS:000318211100007,
Author = {Hewings, David S. and Fedorov, Oleg and Filippakopoulos, Panagis and
Martin, Sarah and Picaud, Sarah and Tumber, Anthony and Wells,
Christopher and Olcina, Monica M. and Freeman, Katherine and Gill,
Andrew and Ritchie, Alison J. and Sheppard, David W. and Russell, Angela
J. and Hammond, Ester M. and Knapp, Stefan and Brennan, Paul E. and
Conway, Stuart J.},
Title = {Optimization of 3,5-Dimethylisoxazole Derivatives as Potent Bromodomain
Ligands},
Journal = {JOURNAL OF MEDICINAL CHEMISTRY},
Year = {2013},
Volume = {56},
Number = {8},
Pages = {3217-3227},
Month = {APR 25},
DOI = {10.1021/jm301588r},
ISSN = {0022-2623},
EISSN = {1520-4804},
ResearcherID-Numbers = {Knapp, Stefan/AAG-2347-2019
Conway, Stuart/AAP-3526-2020
Fedorov, Oleg/B-6412-2014
},
ORCID-Numbers = {Filippakopoulos, Panagis/0000-0002-1515-1317
Knapp, Stefan/0000-0001-5995-6494
Russell, Angela/0000-0003-3610-9369
Conway, Stuart/0000-0002-5148-117X
Hammond, Ester/0000-0002-2335-3146
Hewings, David/0000-0001-9451-8959
Fedorov, Oleg/0000-0001-9004-1815
Wells-Holland, Chris/0000-0001-9985-9816},
Unique-ID = {WOS:000318211100007},
}
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