Generation of a Selective Small Molecule Inhibitor of the CBP/p300 Bromodomain for Leukemia Therapy. Picaud, S., Fedorov, O., Thanasopoulou, A., Leonards, K., Jones, K., Meier, J., Olzscha, H., Monteiro, O., Martin, S., Philpott, M., Tumber, A., Filippakopoulos, P., Yapp, C., Wells, C., Che, K. H., Bannister, A., Robson, S., Kumar, U., Parr, N., Lee, K., Lugo, D., Jeffrey, P., Taylor, S., Vecellio, M. L., Bountra, C., Brennan, P. E., O'Mahony, A., Velichko, S., Mueller, S., Hay, D., Daniels, D. L., Urh, M., La Thangue, N. B., Kouzarides, T., Prinjha, R., Schwaller, J., & Knapp, S. CANCER RESEARCH, 75(23):5106-5119, DEC 1, 2015.
doi  bibtex   
@article{ WOS:000365603000011,
Author = {Picaud, Sarah and Fedorov, Oleg and Thanasopoulou, Angeliki and
   Leonards, Katharina and Jones, Katherine and Meier, Julia and Olzscha,
   Heidi and Monteiro, Octovia and Martin, Sarah and Philpott, Martin and
   Tumber, Anthony and Filippakopoulos, Panagis and Yapp, Clarence and
   Wells, Christopher and Che, Ka Hing and Bannister, Andrew and Robson,
   Samuel and Kumar, Umesh and Parr, Nigel and Lee, Kevin and Lugo, Dave
   and Jeffrey, Philip and Taylor, Simon and Vecellio, Matteo L. and
   Bountra, Chas and Brennan, Paul E. and O'Mahony, Alison and Velichko,
   Sharlene and Mueller, Susanne and Hay, Duncan and Daniels, Danette L.
   and Urh, Marjeta and La Thangue, Nicholas B. and Kouzarides, Tony and
   Prinjha, Rab and Schwaller, Juerg and Knapp, Stefan},
Title = {Generation of a Selective Small Molecule Inhibitor of the CBP/p300
   Bromodomain for Leukemia Therapy},
Journal = {CANCER RESEARCH},
Year = {2015},
Volume = {75},
Number = {23},
Pages = {5106-5119},
Month = {DEC 1},
DOI = {10.1158/0008-5472.CAN-15-0236},
ISSN = {0008-5472},
EISSN = {1538-7445},
ResearcherID-Numbers = {Knapp, Stefan/AAG-2347-2019
   Olzscha, Heidi/AAU-1296-2020
   Vecellio, Matteo Luca/HGB-6768-2022
   Schwaller, Juerg/A-3044-2016
   Fedorov, Oleg/B-6412-2014
   Brown, Tom/A-6655-2010
   },
ORCID-Numbers = {Knapp, Stefan/0000-0001-5995-6494
   Philpott, Martin/0000-0003-3632-0084
   Muller-Knapp, Susanne/0000-0003-2402-4157
   Brennan, Paul/0000-0002-8950-7646
   Robson, Samuel Charles/0000-0001-5702-9160
   Vecellio, Matteo Luca/0000-0002-8643-1316
   Bannister, Andrew/0000-0002-6312-4436
   Filippakopoulos, Panagis/0000-0002-1515-1317
   Kouzarides, Tony/0000-0002-8918-4162
   Olzscha, Heidi/0000-0002-1929-1384},
Unique-ID = {WOS:000365603000011},
}

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