RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. Picaud, S., Wells, C., Felletar, I., Brotherton, D., Martin, S., Savitsky, P., Diez-Dacal, B., Philpott, M., Bountra, C., Lingard, H., Fedorov, O., Mueller, S., Brennan, P. E., Knapp, S., & Filippakopoulos, P. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 110(49):19754-19759, DEC 3, 2013.
doi  bibtex   
@article{ WOS:000327744900034,
Author = {Picaud, Sarah and Wells, Christopher and Felletar, Ildiko and
   Brotherton, Deborah and Martin, Sarah and Savitsky, Pavel and
   Diez-Dacal, Beatriz and Philpott, Martin and Bountra, Chas and Lingard,
   Hannah and Fedorov, Oleg and Mueller, Susanne and Brennan, Paul E. and
   Knapp, Stefan and Filippakopoulos, Panagis},
Title = {RVX-208, an inhibitor of BET transcriptional regulators with selectivity
   for the second bromodomain},
Journal = {PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF
   AMERICA},
Year = {2013},
Volume = {110},
Number = {49},
Pages = {19754-19759},
Month = {DEC 3},
DOI = {10.1073/pnas.1310658110},
ISSN = {0027-8424},
ResearcherID-Numbers = {Brown, Tom/A-6655-2010
   Knapp, Stefan/AAG-2347-2019
   Fedorov, Oleg/B-6412-2014
   },
ORCID-Numbers = {Lingard, Hannah/0000-0003-2571-2496
   Filippakopoulos, Panagis/0000-0002-1515-1317
   Brennan, Paul/0000-0002-8950-7646
   Savitsky, Pavel/0000-0001-8584-7750
   Knapp, Stefan/0000-0001-5995-6494
   Wells-Holland, Chris/0000-0001-9985-9816
   Fedorov, Oleg/0000-0001-9004-1815
   Philpott, Martin/0000-0003-3632-0084
   Muller-Knapp, Susanne/0000-0003-2402-4157},
Unique-ID = {WOS:000327744900034},
}

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