RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. Picaud, S., Wells, C., Felletar, I., Brotherton, D., Martin, S., Savitsky, P., Diez-Dacal, B., Philpott, M., Bountra, C., Lingard, H., Fedorov, O., Mueller, S., Brennan, P. E., Knapp, S., & Filippakopoulos, P. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 110(49):19754-19759, DEC 3, 2013. doi bibtex @article{ WOS:000327744900034,
Author = {Picaud, Sarah and Wells, Christopher and Felletar, Ildiko and
Brotherton, Deborah and Martin, Sarah and Savitsky, Pavel and
Diez-Dacal, Beatriz and Philpott, Martin and Bountra, Chas and Lingard,
Hannah and Fedorov, Oleg and Mueller, Susanne and Brennan, Paul E. and
Knapp, Stefan and Filippakopoulos, Panagis},
Title = {RVX-208, an inhibitor of BET transcriptional regulators with selectivity
for the second bromodomain},
Journal = {PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF
AMERICA},
Year = {2013},
Volume = {110},
Number = {49},
Pages = {19754-19759},
Month = {DEC 3},
DOI = {10.1073/pnas.1310658110},
ISSN = {0027-8424},
ResearcherID-Numbers = {Brown, Tom/A-6655-2010
Knapp, Stefan/AAG-2347-2019
Fedorov, Oleg/B-6412-2014
},
ORCID-Numbers = {Lingard, Hannah/0000-0003-2571-2496
Filippakopoulos, Panagis/0000-0002-1515-1317
Brennan, Paul/0000-0002-8950-7646
Savitsky, Pavel/0000-0001-8584-7750
Knapp, Stefan/0000-0001-5995-6494
Wells-Holland, Chris/0000-0001-9985-9816
Fedorov, Oleg/0000-0001-9004-1815
Philpott, Martin/0000-0003-3632-0084
Muller-Knapp, Susanne/0000-0003-2402-4157},
Unique-ID = {WOS:000327744900034},
}
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