A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation-π Interaction. Rooney, T. P. C., Filippakopoulos, P., Fedorov, O., Picaud, S., Cortopassi, W. A., Hay, D. A., Martin, S., Tumber, A., Rogers, C. M., Philpott, M., Wang, M., Thompson, A. L., Heightman, T. D., Pryde, D. C., Cook, A., Paton, R. S., Mueller, S., Knapp, S., Brennan, P. E., & Conway, S. J. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 53(24):6126-6130, JUN, 2014.
doi  bibtex   
@article{ WOS:000337095000015,
Author = {Rooney, Timothy P. C. and Filippakopoulos, Panagis and Fedorov, Oleg and
   Picaud, Sarah and Cortopassi, Wilian A. and Hay, Duncan A. and Martin,
   Sarah and Tumber, Anthony and Rogers, Catherine M. and Philpott, Martin
   and Wang, Minghua and Thompson, Amber L. and Heightman, Tom D. and
   Pryde, David C. and Cook, Andrew and Paton, Robert S. and Mueller,
   Susanne and Knapp, Stefan and Brennan, Paul E. and Conway, Stuart J.},
Title = {A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit
   Pocket Stabilized by a Cation-π Interaction},
Journal = {ANGEWANDTE CHEMIE-INTERNATIONAL EDITION},
Year = {2014},
Volume = {53},
Number = {24},
Pages = {6126-6130},
Month = {JUN},
DOI = {10.1002/anie.201402750},
ISSN = {1433-7851},
EISSN = {1521-3773},
ResearcherID-Numbers = {Knapp, Stefan/AAG-2347-2019
   Conway, Stuart/AAP-3526-2020
   Cook, Andrew/A-8652-2015
   Paton, Robert/A-4564-2010
   Brown, Tom/A-6655-2010
   Cortopassi, Wilian/P-3136-2014
   },
ORCID-Numbers = {Filippakopoulos, Panagis/0000-0002-1515-1317
   Rooney, Timothy/0000-0001-6788-5526
   Conway, Stuart/0000-0002-5148-117X
   Philpott, Martin/0000-0003-3632-0084
   Brennan, Paul/0000-0002-8950-7646
   Muller-Knapp, Susanne/0000-0003-2402-4157
   Cortopassi, Wilian/0000-0001-8038-7847
   Knapp, Stefan/0000-0001-5995-6494
   Paton, Robert/0000-0002-0104-4166},
Unique-ID = {WOS:000337095000015},
}

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