A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation-π Interaction. Rooney, T. P. C., Filippakopoulos, P., Fedorov, O., Picaud, S., Cortopassi, W. A., Hay, D. A., Martin, S., Tumber, A., Rogers, C. M., Philpott, M., Wang, M., Thompson, A. L., Heightman, T. D., Pryde, D. C., Cook, A., Paton, R. S., Mueller, S., Knapp, S., Brennan, P. E., & Conway, S. J. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 53(24):6126-6130, JUN, 2014. doi bibtex @article{ WOS:000337095000015,
Author = {Rooney, Timothy P. C. and Filippakopoulos, Panagis and Fedorov, Oleg and
Picaud, Sarah and Cortopassi, Wilian A. and Hay, Duncan A. and Martin,
Sarah and Tumber, Anthony and Rogers, Catherine M. and Philpott, Martin
and Wang, Minghua and Thompson, Amber L. and Heightman, Tom D. and
Pryde, David C. and Cook, Andrew and Paton, Robert S. and Mueller,
Susanne and Knapp, Stefan and Brennan, Paul E. and Conway, Stuart J.},
Title = {A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit
Pocket Stabilized by a Cation-π Interaction},
Journal = {ANGEWANDTE CHEMIE-INTERNATIONAL EDITION},
Year = {2014},
Volume = {53},
Number = {24},
Pages = {6126-6130},
Month = {JUN},
DOI = {10.1002/anie.201402750},
ISSN = {1433-7851},
EISSN = {1521-3773},
ResearcherID-Numbers = {Knapp, Stefan/AAG-2347-2019
Conway, Stuart/AAP-3526-2020
Cook, Andrew/A-8652-2015
Paton, Robert/A-4564-2010
Brown, Tom/A-6655-2010
Cortopassi, Wilian/P-3136-2014
},
ORCID-Numbers = {Filippakopoulos, Panagis/0000-0002-1515-1317
Rooney, Timothy/0000-0001-6788-5526
Conway, Stuart/0000-0002-5148-117X
Philpott, Martin/0000-0003-3632-0084
Brennan, Paul/0000-0002-8950-7646
Muller-Knapp, Susanne/0000-0003-2402-4157
Cortopassi, Wilian/0000-0001-8038-7847
Knapp, Stefan/0000-0001-5995-6494
Paton, Robert/0000-0002-0104-4166},
Unique-ID = {WOS:000337095000015},
}
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C. and Filippakopoulos, Panagis and Fedorov, Oleg and\n Picaud, Sarah and Cortopassi, Wilian A. and Hay, Duncan A. and Martin,\n Sarah and Tumber, Anthony and Rogers, Catherine M. and Philpott, Martin\n and Wang, Minghua and Thompson, Amber L. and Heightman, Tom D. and\n Pryde, David C. and Cook, Andrew and Paton, Robert S. and Mueller,\n Susanne and Knapp, Stefan and Brennan, Paul E. and Conway, Stuart J.},\nTitle = {A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit\n Pocket Stabilized by a Cation-π Interaction},\nJournal = {ANGEWANDTE CHEMIE-INTERNATIONAL EDITION},\nYear = {2014},\nVolume = {53},\nNumber = {24},\nPages = {6126-6130},\nMonth = {JUN},\nDOI = {10.1002/anie.201402750},\nISSN = {1433-7851},\nEISSN = {1521-3773},\nResearcherID-Numbers = {Knapp, Stefan/AAG-2347-2019\n Conway, Stuart/AAP-3526-2020\n Cook, Andrew/A-8652-2015\n Paton, Robert/A-4564-2010\n Brown, Tom/A-6655-2010\n Cortopassi, Wilian/P-3136-2014\n },\nORCID-Numbers = {Filippakopoulos, Panagis/0000-0002-1515-1317\n Rooney, Timothy/0000-0001-6788-5526\n Conway, Stuart/0000-0002-5148-117X\n Philpott, Martin/0000-0003-3632-0084\n Brennan, Paul/0000-0002-8950-7646\n Muller-Knapp, Susanne/0000-0003-2402-4157\n Cortopassi, Wilian/0000-0001-8038-7847\n Knapp, Stefan/0000-0001-5995-6494\n Paton, Robert/0000-0002-0104-4166},\nUnique-ID = {WOS:000337095000015},\n}\n\n","author_short":["Rooney, T. 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