Discovery of novel benzothiophene derivatives as potent and narrow spectrum inhibitors of DYRK1A and DYRK1B

Discovery of novel benzothiophene derivatives as potent and narrow spectrum inhibitors of DYRK1A and DYRK1B. Segretti, N. D., Takarada, J. E., Ferreira, M. A., Da Silva Santiago, A., Teodoro, B. V., Damião, M. C., Godoi, P. H., Cunha, M. R., Fala, A. M., Ramos, P. Z., Ishikawa, E. E., Mascarello, A., Serafim, R. A., Azevedo, H., Guimarães, C. R., & Couñago, R. M. Bioorganic & Medicinal Chemistry Letters, 68:128764, July, 2022.

Paper doi bibtex

@article{segretti_discovery_2022,
	title = {Discovery of novel benzothiophene derivatives as potent and narrow spectrum inhibitors of {DYRK1A} and {DYRK1B}},
	volume = {68},
	copyright = {Licença Creative Commons Attribution-NonCommercial-NoDerivatives 4.0 International},
	issn = {0960894X},
	url = {https://linkinghub.elsevier.com/retrieve/pii/S0960894X22002402},
	doi = {10.1016/j.bmcl.2022.128764},
	language = {en},
	urldate = {2026-02-08},
	journal = {Bioorganic \& Medicinal Chemistry Letters},
	author = {Segretti, Natanael D. and Takarada, Jéssica E. and Ferreira, Marcos A. and Da Silva Santiago, André and Teodoro, Bruno V.M. and Damião, Mariana C.F.C.B. and Godoi, Paulo H. and Cunha, Micael R. and Fala, Angela M. and Ramos, Priscila Z. and Ishikawa, Eloisa E. and Mascarello, Alessandra and Serafim, Ricardo A.M. and Azevedo, Hatylas and Guimarães, Cristiano R.W. and Couñago, Rafael M.},
	month = jul,
	year = {2022},
	pages = {128764},
}

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