Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells. Tumber, A., Nuzzi, A., Hookway, E. S., Hatch, S. B., Velupillai, S., Johansson, C., Kawamura, A., Savitsky, P., Yapp, C., Szykowska, A., Wu, N., Bountra, C., Strain-Damerell, C., Burgess-Brown, N. A., Ruda, G. F., Fedorov, O., Munro, S., England, K. S., Nowak, R. P., Schofield, C. J., La Thangue, N. B., Pawlyn, C., Davies, F., Morgan, G., Athanasou, N., Mueller, S., Oppermann, U., & Brennan, P. E. CELL CHEMICAL BIOLOGY, 24(3):371-380, MAR 16, 2017. doi bibtex @article{ WOS:000397424600014,
Author = {Tumber, Anthony and Nuzzi, Andrea and Hookway, Edward S. and Hatch,
Stephanie B. and Velupillai, Srikannathasan and Johansson, Catrine and
Kawamura, Akane and Savitsky, Pavel and Yapp, Clarence and Szykowska,
Aleksandra and Wu, Na and Bountra, Chas and Strain-Damerell, Claire and
Burgess-Brown, Nicola A. and Ruda, Gian Filippo and Fedorov, Oleg and
Munro, Shonagh and England, Katherine S. and Nowak, Radoslaw P. and
Schofield, Christopher J. and La Thangue, Nicholas B. and Pawlyn,
Charlotte and Davies, Faith and Morgan, Gareth and Athanasou, Nick and
Mueller, Susanne and Oppermann, Udo and Brennan, Paul E.},
Title = {Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of
H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma
Cells},
Journal = {CELL CHEMICAL BIOLOGY},
Year = {2017},
Volume = {24},
Number = {3},
Pages = {371-380},
Month = {MAR 16},
DOI = {10.1016/j.chembiol.2017.02.006},
ISSN = {2451-9448},
ResearcherID-Numbers = {Fedorov, Oleg/A-3201-2019
Morgan, Gareth/G-3603-2010
Hookway, Edward/I-2613-2018
Nowak, Radosław/JLM-2338-2023
Knapp, Stefan/AAG-2347-2019
Kawamura, Akane/I-4047-2018
},
ORCID-Numbers = {England, Katherine/0000-0002-4921-7505
Schofield, Christopher/0000-0002-0290-6565
Fedorov, Oleg/0000-0001-5268-6399
Hatch, Stephanie/0000-0002-7401-9279
Pawlyn, Charlotte/0000-0002-7190-0028
Davies, Faith/0000-0002-3971-2393
Schofield, Chris/0009-0008-4988-0199
Savitsky, Pavel/0000-0001-8584-7750
Kawamura, Akane/0000-0003-1169-5082
Brennan, Paul/0000-0002-8950-7646
Muller-Knapp, Susanne/0000-0003-2402-4157
morgan, gareth/0000-0002-4271-6360
Ruda, Gian Filippo/0000-0001-6150-2715
Nowak, Radoslaw/0000-0002-0605-0071},
Unique-ID = {WOS:000397424600014},
}
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