Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells. Tumber, A., Nuzzi, A., Hookway, E. S., Hatch, S. B., Velupillai, S., Johansson, C., Kawamura, A., Savitsky, P., Yapp, C., Szykowska, A., Wu, N., Bountra, C., Strain-Damerell, C., Burgess-Brown, N. A., Ruda, G. F., Fedorov, O., Munro, S., England, K. S., Nowak, R. P., Schofield, C. J., La Thangue, N. B., Pawlyn, C., Davies, F., Morgan, G., Athanasou, N., Mueller, S., Oppermann, U., & Brennan, P. E. CELL CHEMICAL BIOLOGY, 24(3):371-380, MAR 16, 2017.
doi  bibtex   
@article{ WOS:000397424600014,
Author = {Tumber, Anthony and Nuzzi, Andrea and Hookway, Edward S. and Hatch,
   Stephanie B. and Velupillai, Srikannathasan and Johansson, Catrine and
   Kawamura, Akane and Savitsky, Pavel and Yapp, Clarence and Szykowska,
   Aleksandra and Wu, Na and Bountra, Chas and Strain-Damerell, Claire and
   Burgess-Brown, Nicola A. and Ruda, Gian Filippo and Fedorov, Oleg and
   Munro, Shonagh and England, Katherine S. and Nowak, Radoslaw P. and
   Schofield, Christopher J. and La Thangue, Nicholas B. and Pawlyn,
   Charlotte and Davies, Faith and Morgan, Gareth and Athanasou, Nick and
   Mueller, Susanne and Oppermann, Udo and Brennan, Paul E.},
Title = {Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of
   H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma
   Cells},
Journal = {CELL CHEMICAL BIOLOGY},
Year = {2017},
Volume = {24},
Number = {3},
Pages = {371-380},
Month = {MAR 16},
DOI = {10.1016/j.chembiol.2017.02.006},
ISSN = {2451-9448},
ResearcherID-Numbers = {Fedorov, Oleg/A-3201-2019
   Morgan, Gareth/G-3603-2010
   Hookway, Edward/I-2613-2018
   Nowak, Radosław/JLM-2338-2023
   Knapp, Stefan/AAG-2347-2019
   Kawamura, Akane/I-4047-2018
   },
ORCID-Numbers = {England, Katherine/0000-0002-4921-7505
   Schofield, Christopher/0000-0002-0290-6565
   Fedorov, Oleg/0000-0001-5268-6399
   Hatch, Stephanie/0000-0002-7401-9279
   Pawlyn, Charlotte/0000-0002-7190-0028
   Davies, Faith/0000-0002-3971-2393
   Schofield, Chris/0009-0008-4988-0199
   Savitsky, Pavel/0000-0001-8584-7750
   Kawamura, Akane/0000-0003-1169-5082
   Brennan, Paul/0000-0002-8950-7646
   Muller-Knapp, Susanne/0000-0003-2402-4157
   morgan, gareth/0000-0002-4271-6360
   Ruda, Gian Filippo/0000-0001-6150-2715
   Nowak, Radoslaw/0000-0002-0605-0071},
Unique-ID = {WOS:000397424600014},
}

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