Design, Synthesis and Characterization of Covalent KDM5 Inhibitors. Vazquez-Rodriguez, S., Wright, M., Rogers, C. M., Cribbs, A. P., Velupillai, S., Philpott, M., Lee, H., Dunford, J. E., Huber, K. V. M., Robers, M. B., Vasta, J. D., Thezenas, M., Bonham, S., Kessler, B., Bennett, J., Fedorov, O., Raynaud, F., Donovan, A., Blagg, J., Bavetsias, V., Oppermann, U., Bountra, C., Kawamura, A., & Brennan, P. E. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 58(2):515-519, JAN 8, 2019.
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@article{ WOS:000454944900022,
Author = {Vazquez-Rodriguez, Saleta and Wright, Miranda and Rogers, Catherine M.
   and Cribbs, Adam P. and Velupillai, Srikannathasan and Philpott, Martin
   and Lee, Henry and Dunford, James E. and Huber, Kilian V. M. and Robers,
   Matthew B. and Vasta, James D. and Thezenas, Marie-Laetitia and Bonham,
   Sarah and Kessler, Benedikt and Bennett, James and Fedorov, Oleg and
   Raynaud, Florence and Donovan, Adam and Blagg, Julian and Bavetsias,
   Vassilios and Oppermann, Udo and Bountra, Chas and Kawamura, Akane and
   Brennan, Paul E.},
Title = {Design, Synthesis and Characterization of Covalent KDM5 Inhibitors},
Journal = {ANGEWANDTE CHEMIE-INTERNATIONAL EDITION},
Year = {2019},
Volume = {58},
Number = {2},
Pages = {515-519},
Month = {JAN 8},
DOI = {10.1002/anie.201810179},
ISSN = {1433-7851},
EISSN = {1521-3773},
ResearcherID-Numbers = {Cribbs, Adam/U-4055-2019
   Kessler, Benedikt/JGC-6978-2023
   Fedorov, Oleg/A-3201-2019
   Brown, Tom/A-6655-2010
   Kawamura, Akane/I-4047-2018
   Vazquez-Rodriguez, Saleta/L-4047-2014
   Huber, Kilian/L-6921-2015
   },
ORCID-Numbers = {Fedorov, Oleg/0000-0001-5268-6399
   Kessler, Benedikt/0000-0002-8160-2446
   Vazquez-Rodriguez, Saleta/0000-0003-1356-8984
   Huber, Kilian/0000-0002-1103-5300
   Cribbs, Adam/0000-0001-5288-3077
   Brennan, Paul/0000-0002-8950-7646
   Philpott, Martin/0000-0003-3632-0084
   Dunford, James/0000-0002-9932-4042
   Raynaud, Florence/0000-0003-0957-6279
   Bennett, James/0000-0003-1396-8400},
Unique-ID = {WOS:000454944900022},
}

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