Design, Synthesis and Characterization of Covalent KDM5 Inhibitors. Vazquez-Rodriguez, S., Wright, M., Rogers, C., M., Cribbs, A., P., Velupillai, S., Philpott, M., Lee, H., Dunford, J., E., Huber, K., V., M., Robers, M., B., Vasta, J., D., Thezenas, M., Bonham, S., Kessler, B., Bennett, J., Fedorov, O., Raynaud, F., Donovan, A., Blagg, J., Bavetsias, V., Oppermann, U., Bountra, C., Kawamura, A., & Brennan, P., E. Angewandte Chemie International Edition, 58(2):515-519, John Wiley & Sons, Ltd, 1, 2019.
Paper
Website doi bibtex 13 downloads @article{
title = {Design, Synthesis and Characterization of Covalent KDM5 Inhibitors},
type = {article},
year = {2019},
keywords = {KDM5,covalent inhibitors,epigenetics,lysine demethylase},
pages = {515-519},
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citation_key = {Vazquez-Rodriguez2019},
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author = {Vazquez-Rodriguez, Saleta and Wright, Miranda and Rogers, Catherine M. and Cribbs, Adam P. and Velupillai, Srikannathasan and Philpott, Martin and Lee, Henry and Dunford, James E. and Huber, Kilian V. M. and Robers, Matthew B. and Vasta, James D. and Thezenas, Marie-Laetitia and Bonham, Sarah and Kessler, Benedikt and Bennett, James and Fedorov, Oleg and Raynaud, Florence and Donovan, Adam and Blagg, Julian and Bavetsias, Vassilios and Oppermann, Udo and Bountra, Chas and Kawamura, Akane and Brennan, Paul E.},
doi = {10.1002/anie.201810179},
journal = {Angewandte Chemie International Edition},
number = {2}
}
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